Pyridostigmine Controlled-Release Tablets

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Pyridostigmine Controlled-Release Tablets


Generic Name: Pyridostigmine Controlled-Release Tablets (peer-id-oh-STIG-meen)
Brand Name: Mestinon

Pyridostigmine Controlled-Release Tablets is used for:

Treating myasthenia gravis. It may also be used for other conditions as determined by your doctor.

Pyridostigmine Controlled-Release Tablets is a cholinesterase inhibitor. It works by improving nerve impulses in muscles so that the muscles are better able to work.

Do NOT use Pyridostigmine Controlled-Release Tablets if:

  • you are allergic to any ingredient in Pyridostigmine Controlled-Release Tablets
  • you are taking quinine or quinidine
  • you have a stomach, intestinal, or urinary blockage

Contact your doctor or health care provider right away if any of these apply to you.

Before using Pyridostigmine Controlled-Release Tablets:

Some medical conditions may interact with Pyridostigmine Controlled-Release Tablets. Tell your doctor or pharmacist if you have any medical conditions, especially if any of the following apply to you:

  • if you are pregnant, planning to become pregnant, or are breast-feeding
  • if you are taking any prescription or nonprescription medicine, herbal preparation, or dietary supplement
  • if you have allergies to medicines, foods, or other substances
  • if you have heart problems (eg, heart block, slow heartbeat), a urinary tract infection, asthma, or kidney problems

Some MEDICINES MAY INTERACT with Pyridostigmine Controlled-Release Tablets. Tell your health care provider if you are taking any other medicines, especially any of the following:

  • Quinine or quinidine because effectiveness of Pyridostigmine Controlled-Release Tablets may be decreased
  • Succinylcholine because actions and side effects may be increased by Pyridostigmine Controlled-Release Tablets

This may not be a complete list of all interactions that may occur. Ask your health care provider if Pyridostigmine Controlled-Release Tablets may interact with other medicines that you take. Check with your health care provider before you start, stop, or change the dose of any medicine.

How to use Pyridostigmine Controlled-Release Tablets:

Use Pyridostigmine Controlled-Release Tablets as directed by your doctor. Check the label on the medicine for exact dosing instructions.

  • Pyridostigmine Controlled-Release Tablets may be taken with or without food. Take with food if it upsets your stomach.
  • Swallow Pyridostigmine Controlled-Release Tablets whole. Do not break, crush, or chew before swallowing.
  • If you miss a dose of Pyridostigmine Controlled-Release Tablets, take it as soon as possible. If it is almost time for your next dose, skip the missed dose and go back to your regular dosing schedule. Do not take 2 doses at once.

Ask your health care provider any questions you may have about how to use Pyridostigmine Controlled-Release Tablets.

Important safety information:

  • Before you have any medical or dental treatments, emergency care, or surgery, tell the doctor or dentist that you are using Pyridostigmine Controlled-Release Tablets.
  • Use Pyridostigmine Controlled-Release Tablets with extreme caution in CHILDREN. Safety and effectiveness have not been confirmed.
  • PREGNANCY and BREAST-FEEDING: If you become pregnant while taking Pyridostigmine Controlled-Release Tablets, discuss with your doctor the benefits and risks of using Pyridostigmine Controlled-Release Tablets during pregnancy. Pyridostigmine Controlled-Release Tablets is excreted in breast milk. If you are or will be breast-feeding while you are using Pyridostigmine Controlled-Release Tablets, check with your doctor or pharmacist to discuss the risks to your baby.

Possible side effects of Pyridostigmine Controlled-Release Tablets:

All medicines may cause side effects, but many people have no, or minor, side effects. When used in small doses, no COMMON side effects have been reported with this product. Seek medical attention right away if any of these SEVERE side effects occur:

Severe allergic reactions (rash; hives; itching; difficulty breathing; tightness in the chest; swelling of the mouth, face, lips, or tongue); diarrhea; fainting; increased production of saliva; increased sweating; muscle weakness; nausea; small pupils; stomach cramps; trouble breathing; vision changes; vomiting; weakness.

This is not a complete list of all side effects that may occur. If you have questions or need medical advice about side effects, contact your doctor or health care provider. You may report side effects to the FDA at 1-800-FDA-1088 (1-800-332-1088) or at http://www.fda.gov/medwatch.

If OVERDOSE is suspected:

Contact 1-800-222-1222 (the American Association of Poison Control Centers), your local poison control center (http://www.aapcc.org/findyour.htm), or emergency room immediately. Symptoms may include diarrhea; fainting; increased production of saliva; increased sweating; muscle weakness; nausea; small pupils; stomach cramps; trouble breathing; vision changes; vomiting; weakness.

Proper storage of Pyridostigmine Controlled-Release Tablets:

Store Pyridostigmine Controlled-Release Tablets between 68 and 77 degrees F (20 and 25 degrees C). Store away from heat, moisture, and light. Do not store in the bathroom. Keep Pyridostigmine Controlled-Release Tablets out of the reach of children and away from pets.

General information:

  • If you have any questions about Pyridostigmine Controlled-Release Tablets, please talk with your doctor, pharmacist, or other health care provider.
  • Pyridostigmine Controlled-Release Tablets is to be used only by the patient for whom it is prescribed. Do not share it with other people.
  • If your symptoms do not improve or if they become worse, check with your doctor.

This information is a summary only. It does not contain all information about Pyridostigmine Controlled-Release Tablets. If you have questions about the medicine you are taking or would like more information, check with your doctor, pharmacist, or other health care provider.

Issue Date: November 1, 2006
Database Edition 06.4.1.002
Copyright © 2006 Wolters Kluwer Health, Inc.




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