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|Methyltestosterone |
Drugs search, click the first letter of a drug name: | A | B | C | D | E | F | G | H | I | J | K | L | M | N | O | P | Q | R | S | T | U | V | W | X | Y | Z | 1 | 2 | 3 | 4 | 5 | 6 | 8 | 9 Home MethyltestosteronePronouncation: (METH-ill-tess-TAHS-ter-ohn)Class: Androgen Trade Names: Trade Names: Trade Names: Trade Names: Mechanism of ActionPharmacologyPromotes growth and development of male reproductive organs, maintains secondary sex characteristics, increases protein anabolism, and decreases protein catabolism. PharmacokineticsMetabolismBecause methyltestosterone is less extensively metabolized by the liver and has a longer t ½ than testosterone, methyltestosterone is more suitable than testosterone for oral administration. Indications and UsageReplacement therapy in the following conditions associated with a deficiency or absence of endogenous testosterone: primary hypogonadism (congenital or acquired); hypogonadotropic hypogonadism (congenital or acquired); delayed puberty (males); used secondarily in advancing inoperable metastatic (skeletal) mammary cancer (females). ContraindicationsMen with carcinoma of the breast; men with known or suspected carcinoma of the prostate gland; women known or suspected to be pregnant; hypersensitivity to any component of the product. Dosage and AdministrationCongenital or Acquired Primary Hypogonadism, Hypogonadotropic HypogonadismAdults (men) PO 10 to 50 mg/day. Delayed PubertyAdults (men) PO Doses are generally in the lower range of the above doses for hypogonadism and for a limited duration (eg, 4 to 6 mo). Metastatic Breast CarcinomaAdults (women) PO 50 to 200 mg/day. Storage/StabilityStore tablets and capsules at ambient room temperature (59° to 86°F). Protect from light, moisture, and heat. Drug InteractionsInsulinBlood glucose levels may be reduced by methyltestosterone, decreasing insulin requirements. Oral anticoagulants (eg, warfarin)Effects of oral anticoagulant may be increased. Dosage reduction may be required. Laboratory Test InteractionsThyroxine-binding globulin levels may be decreased; however, thyroid hormone levels remain unchanged and there is no clinical evidence of thyroid dysfunction. Adverse ReactionsCNSIncreased and decreased libido; headache; anxiety; depression; generalized paresthesia. DermatologicHirsutism; male pattern baldness; acne. ElectrolytesRetention of sodium, chloride, water, potassium, calcium, and inorganic phosphates. GINausea. GenitourinaryAmenorrhea, menstrual irregularities, inhibition of gonadotropin secretion, virilization (including deepening of voice and clitoral enlargement for women); gynecomastia, excessive frequency and duration of penile erection, oligospermia (men). HematologicSuppression of clotting factors II, V, VII, and X; bleeding in patients with polycythemia. HepaticCholestatic jaundice; alterations in LFTs; hepatocellular neoplasms; peliosis hepatitis. MetabolicIncreased serum cholesterol. MiscellaneousAnaphylactoid reactions. PrecautionsPregnancyCategory X . LactationUndetermined. ChildrenUse with caution and only by specialists aware of the adverse effects on bone maturation. ElderlyElderly men may be at increased risk of developing prostatic hypertrophy or carcinoma. Athletic performanceAbuse of this agent to enhance athletic performance has potential risk of serious side effects. Delayed pubertyBecause bone maturation without producing compensatory linear growth can occur, use with caution in males with delayed puberty. EdemaUse with caution in patients with conditions that might be affected by fluid retention (eg, renal, hepatic, cardiac disease). GynecomastiaMay occur and persist in patients being treated for hypogonadism. Hepatic effectsCholestatic hepatitis and jaundice may occur. Prolonged use of high doses may result in hepatic adenomas, hepatocellular carcinoma, and peliosis hepatitis. HypercalcemiaMay cause hypercalcemia when used in patients with breast cancer. Oligospermia and reduced ejaculatory volumeMay occur after prolonged use. PriapismMay be indicative of excessive dosage. VirilizationMay occur in women using high-dose androgens. Patient Information
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