Enalapril maleate, Felodipine

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Enalapril maleate, Felodipine

Generic name: Enalapril maleate, Felodipine
Brand names: Lexxel

Why is Enalapril maleate, Felodipine prescribed?

Enalapril maleate, Felodipine is used to treat high blood pressure. It combines two blood pressure drugs: an ACE inhibitor and a calcium channel blocker. The ACE inhibitor (enalapril) lowers blood pressure by preventing a chemical in your blood called angiotensin I from converting to a more potent form that narrows the blood vessels and increases salt and water retention. The calcium channel blocker (felodipine) also works to keep the blood vessels open, and eases the heart"s workload by reducing the force and rate of your heartbeat.

Enalapril maleate, Felodipine can be prescribed alone or in combination with other blood pressure medicines, especially water pills (diuretics) such as HydroDIURIL or Esidrix.

Most important fact about Enalapril maleate, Felodipine

Doctors usually prescribe Enalapril maleate, Felodipine for patients who have been taking one of its components--enalapril (Vasotec) or extended-release felodipine (Plendil)--without showing improvement. Like other blood pressure medications, Enalapril maleate, Felodipine must be taken regularly for it to be effective. Since blood pressure declines gradually, it may be 1 or 2 weeks before you get the full benefit of Enalapril maleate, Felodipine; and you must continue taking it even if you are feeling well. Enalapril maleate, Felodipine does not cure high blood pressure; it merely keeps it under control.

How should you take Enalapril maleate, Felodipine?

Enalapril maleate, Felodipine can be taken with a light meal or without food. Remember, however, that a high-fat meal can reduce its effectiveness, and that grapefruit juice increases its impact.

Swallow Enalapril maleate, Felodipine tablets whole. Do not crush, divide, or chew them.

--If you miss a dose...

Take it as soon as you remember. If it is almost time for your next dose, skip the one you missed and go back to your regular schedule. Never take 2 doses at the same time.

--Storage instructions...

Store at room temperature. Keep the container tightly closed and protect from light and humidity.

What side effects may occur?

Side effects cannot be anticipated. If any develop or change in intensity, inform your doctor as soon as possible. Only your doctor can determine if it is safe for you to continue taking Enalapril maleate, Felodipine.

  • More common side effects may include:
    Dizziness, headache, swelling

Why should Enalapril maleate, Felodipine not be prescribed?

Avoid Enalapril maleate, Felodipine if you have ever had an allergic reaction to it, or have ever developed a swollen throat and difficulty swallowing (angioedema) while taking similar drugs such as Capoten, Vasotec, or Zestril. Make sure your doctor is aware of the incident.

Special warnings about Enalapril maleate, Felodipine

Call your doctor immediately if you begin to suffer angioedema while taking Enalapril maleate, Felodipine. Warning signs include swelling of the face, lips, tongue, or throat; swelling of the arms and legs; and difficulty swallowing or breathing.

Bee or wasp venom given to prevent an allergic reaction to stings may cause a severe allergic reaction to Enalapril maleate, Felodipine. Kidney dialysis can also prompt an allergic reaction to the drug.

Enalapril maleate, Felodipine sometimes causes a severe drop in blood pressure. The danger is especially great if you have been taking water pills (diuretics), or if you have heart disease, kidney disease, or a potassium or salt imbalance. Excessive sweating, severe diarrhea, and vomiting are also a threat. They can rob the body of water, causing a dangerous drop in blood pressure. If you feel light-headed or faint, have chest pain, or feel your heart racing, contact your doctor immediately.

Because another of the ACE inhibitors, Capoten, has been known to cause serious blood disorders, your doctor will check your blood regularly while you are taking Enalapril maleate, Felodipine. If you develop signs of infection such as a sore throat or a fever, you should contact your doctor at once--an infection could be a signal of blood abnormalities.

Enalapril maleate, Felodipine may also affect the liver; and your doctor will need to adjust your dosage with extra care if you are over 65 or have liver disease. Report these symptoms of liver problems to your doctor immediately: a generally run-down feeling, pain in the upper right abdomen, or yellowing of the skin or the whites of your eyes.

If you suffer from heart failure or kidney disease, make certain that your doctor knows about it. Enalapril maleate, Felodipine should be used with caution under these circumstances.

Some people taking Enalapril maleate, Felodipine develop a dry, nagging cough. This will go away when you stop taking the drug. Others are troubled by swollen gums. Good dental hygiene makes this less likely.

Possible food and drug interactions when taking Enalapril maleate, Felodipine

If Enalapril maleate, Felodipine is taken with certain other drugs, the effects of either could be increased, decreased, or altered. It is especially important to check with your doctor before combining Enalapril maleate, Felodipine with the following:

Cimetidine (Tagamet)
Diuretics such as Lasix or HydroDIURIL
Diuretics that leave potassium in the body, such as Aldactone, Midamor, and Dyrenium
Epilepsy medications such as Dilantin, phenobarbital, and Tegretol
Erythromycin (E.E.S., E-Mycin, ERYC, others)
Grapefruit juice
High-fat meals
Itraconazole (Sporanox)
Lithium (Eskalith, Lithobid)
Potassium supplements such as K-Lyte, K-Tabs, and Slow-K

Because Enalapril maleate, Felodipine tends to increase your potassium level, avoid potassium-containing salt substitutes unless your doctor approves.

Special information if you are pregnant or breastfeeding

Do not take Enalapril maleate, Felodipine during pregnancy. When taken during the final 6 months, the ACE inhibitor in Enalapril maleate, Felodipine can cause birth defects, prematurity, and death in the developing or newborn baby. If you are pregnant, inform your doctor immediately.

Enalapril maleate, Felodipine may appear in breast milk and could affect a nursing infant. If Enalapril maleate, Felodipine is essential to your health, your doctor may advise you to stop breastfeeding.

Recommended dosage

ADULTS

Enalapril maleate, Felodipine is available in two strengths. Enalapril maleate, Felodipine 5-2.5 contains 5 milligrams of enalapril and 2.5 milligrams of felodipine. Enalapril maleate, Felodipine 5-5 contains 5 milligrams of each.

The usual starting dose is 1 tablet of Enalapril maleate, Felodipine 5-5 once a day. If there is no change in your blood pressure after 1 or 2 weeks, the doctor may increase your dose to 2 tablets once a day. If your blood pressure still remains too high, the dose may be increased to 4 tablets of Enalapril maleate, Felodipine once a day. The doctor may also add a water pill (containing a thiazide) to your regimen.

CHILDREN

The safety and effectiveness of Enalapril maleate, Felodipine in children have not been established.

OLDER ADULTS

If you are over 65, your doctor may have to monitor your blood pressure closely at the beginning of treatment, and adjust your dose with care.

Overdosage

Any medication taken in excess can have serious consequences. If you suspect an overdose, seek medical treatment immediately.

  • Symptoms of Enalapril maleate, Felodipine overdose may include:
    Low blood pressure, rapid heartbeat




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