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|Diazoxide, Parenteral |
Drugs search, click the first letter of a drug name: | A | B | C | D | E | F | G | H | I | J | K | L | M | N | O | P | Q | R | S | T | U | V | W | X | Y | Z | 1 | 2 | 3 | 4 | 5 | 6 | 8 | 9 Home Diazoxide, ParenteralPronouncation: (DIE-aze-OX-ide)Class: Agent for hypertensive emergencies Trade Names: Mechanism of ActionPharmacologyRelaxes smooth muscle in peripheral arterioles, thus reducing BP. PharmacokineticsDistributionGreater than 90% protein bound. Crosses placenta. Eliminationt ½ approximately 28 hr. Onset1 min. Peak2 to 5 min. DurationLess than 12 hr. Indications and UsageShort-term emergency reduction of BP in severe, nonmalignant, and malignant hypertension in hospitalized patients. ContraindicationsDissecting aortic aneurysm; hypersensitivity to thiazides or other sulfonamide derivatives; treatment of compensatory hypertension, such as that associated with aortic coarctation or arteriovenous shunt. Diazoxide is ineffective against hypertension caused by pheochromocytoma. Dosage and AdministrationAdultsIV 1 to 3 mg/kg (max 150 mg in single injection) by rapid injection (no longer than 30 sec). May repeat at 5 to 15 min intervals until satisfactory reduction in BP. May repeat at intervals of 4 to 24 hr until oral therapy can be initiated. Do not use for longer than 10 days. Have patient remain supine during IV administration. Storage/StabilityProtect from light/freezing. Store between 2° to 30°C (36° to 86°F). Drug InteractionsAntihypertensive agentsEnhanced antihypertensive effect. Highly protein-bound agentsHigher blood levels of these agents may occur as a result of displacement by diazoxide. HydantoinsPossible loss of seizure control. SulfonylureasHyperglycemia may occur. Thiazide diureticsMay increase hyperuricemic, hyperglycemic, and antihypertensive effects of diazoxide. Laboratory Test InteractionsHyperglycemia and hyperuricemia produced by diazoxide may affect assessment of these metabolic states. Increased renin secretion and IgG concentrations and decreased cortisol secretion may occur. May cause false-negative insulin response to glucagon. Adverse ReactionsCardiovascularSodium and water retention; hypotension to shock levels; CHF; edema; myocardial ischemia (eg, angina, arrhythmias, ECG changes); supraventricular tachycardia; palpitations; bradycardia. CNSDizziness; weakness; cerebral ischemia; cerebral infarction (eg, unconsciousness, convulsions, paralysis, confusion, focal neurologic deficit); sweating; flushing and feelings of warmth; transient neurologic findings (eg, headache, lethargy, somnolence, euphoria, ringing in the ears, momentary hearing loss). DermatologicCellulitis or phlebitis at site of extravasation; warmth or pain along course of injected vein. GINausea; vomiting; acute pancreatitis (rare); diarrhea; abdominal discomfort. MetabolicHyperglycemia; hyperosmolar coma; hyperuricemia. MiscellaneousHypersensitivity reactions; papilledema. PrecautionsPregnancyCategory C . LactationUndetermined. Special Risk PatientsDiabetic patients may need treatment for hyperglycemia. Use with care in patients with impaired cerebral or cardiac circulation in whom rapid reduction in BP might be deleterious. Observe caution when reducing severely elevated BP. Fluid and electrolyte balanceBecause of sodium and water retention, with possible edema and CHF, concomitant use of diuretic may be needed. However, thiazide diuretics may potentiate diazoxide"s antihypertensive, hyperglycemic, and hyperuricemic actions. OverdosageSymptomsHypotension, hyperglycemia. Patient Information
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