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|Tetracycline Hydrochloride |
Drugs search, click the first letter of a drug name: | A | B | C | D | E | F | G | H | I | J | K | L | M | N | O | P | Q | R | S | T | U | V | W | X | Y | Z | 1 | 2 | 3 | 4 | 5 | 6 | 8 | 9 Home Tetracycline HydrochloridePronouncation: (teh-truh-SIGH-kleen HIGH-droe-KLOR-ide)Class: Anti-infective agent Trade Names: Trade Names: Trade Names: Novo-Tetra (Canada) Nu-Tetra (Canada) Mechanism of ActionPharmacologyInhibits bacterial protein synthesis. PharmacokineticsAbsorptionTetracycline is adequately, but incompletely, absorbed from the GI tract. DistributionTetracycline is about 65% bound to plasma proteins (short-acting). The protein binding for intermediate and long-acting analogs is usually greater. Penetration into most body fluids and tissues is excellent. Tetracycline is distributed in varying degrees in liver, bile, lung, kidney, prostate, urine, CSF, synovial fluid, mucosa of the maxillary sinus, brain, sputum, and bone. Tetracycline crosses the placenta and enters fetal circulation and amniotic fluid. MetabolismTetracycline is concentrated by the liver in the bile. EliminationTetracycline is excreted in both urine and feces at high concentrations in a biologically active form. Special PopulationsRenal Function ImpairmentBecause renal Cl is by glomerular filtration, excretion is significantly affected by the state of renal function. Indications and UsageTreatment of infections caused by susceptible strains of gram-positive and gram-negative bacteria; treatment of Rickettsia , Mycoplasma pneumoniae ; chlamydial infections including treatment of trachoma; adjunctive treatment in severe acne; treatment of susceptible infections when penicillins are contraindicated; adjunctive treatment of acute intestinal amebiasis; treatment of nongonococcal urethritis caused by Ureaplasma urealyticum ; treatment of relapsing fever due to Borrelia recurrentis . ContraindicationsHypersensitivity to tetracyclines or any component. Dosage and AdministrationAdultsPO Usual dose: 1 to 2 g/day in 2 or 4 equal doses. Mild to Moderate Infections500 mg bid or 250 mg qid. Severe Infections500 mg qid. Children older than 8 yr of agePO 25 to 50 mg/kg/day in 4 equally divided doses. BrucellosisAdults PO 500 mg qid for 3 wk, accompanied by 1 g streptomycin IM bid the first week and daily the second week. Severe AcneAdults PO Start with 1 g/day in divided doses; for maintenance, 125 to 500 mg/day (alternate-day or intermittent therapy may be adequate in some patients). Streptococcal InfectionsTreat streptococcal infections for at least 10 days. SyphilisAdults PO Sumycin only: Total dose of 30 to 40 g in equally divided doses over 10 to 15 days. All except Sumycin : Early (less than 1 yr duration) - 500 mg qid for 15 days. More than 1 yr duration - 500 mg qid for 30 days. CDC-recommended treatment for penicillin-allergic patients: Early (less than 1 yr duration) - 500 mg qid for 14 days. More than 1 yr duration - 500 mg qid for 28 days. Uncomplicated GonorrheaAdults PO 500 mg q 6 hr for 7 days. Uncomplicated Urethral, Endocervical, or Rectal Infections Caused by Chlamydia trachomatisAdults PO 500 mg qid for at least 7 days. Storage/StabilityStore capsules, tablets, and oral suspension at controlled room temperature (59° to 86°F). Protect from light and excessive heat. Drug InteractionsAntacids (containing aluminum, calcium, and magnesium), dairy products, food, iron saltsMay decrease oral absorption of tetracycline. AnticoagulantsThe action of oral anticoagulants may be increased. MethoxyfluraneIncreased potential for nephrotoxicity exists; do not use together. Oral contraceptivesMay reduce effect of oral contraceptives. PenicillinsMay interfere with bactericidal action of penicillins. Laboratory Test InteractionsNone well documented. Adverse ReactionsCardiovascularPericarditis (as component of hypersensitivity reaction). CNSDizziness; headache. DermatologicRash; photosensitivity. GIDiarrhea; nausea; vomiting; abdominal pain or discomfort; bulky, loose stools; sore throat; glossitis; anorexia; stomatitis; black hairy tongue; dysphagia; hoarseness; enterocolitis; inflammatory lesions; epigastric distress. GenitourinaryIncreased BUN. HematologicHemolytic anemia; thrombocytopenia; neutropenia; anemia; thrombocytopenic purpura; eosinophilia. MiscellaneousHypersensitivity, including anaphylaxis. PrecautionsPregnancyCategory D . Avoid during pregnancy. LactationExcreted in breast milk. ChildrenAvoid in children younger than 8 yr of age because abnormal bone formation and discoloration of teeth may occur. Renal FunctionExcessive accumulation may occur in patients with renal impairment, resulting in possible liver toxicity; dosage reduction may be required. SuperinfectionProlonged use may result in bacterial or fungal overgrowth. Ophthalmic useMay retard corneal epithelial healing. Outdated productDo not use because degradation products are highly nephrotoxic. Pseudomembranous colitisConsider in patients in whom diarrhea develops. Pseudotumor cerebri (benign intracranial hypertension)Reported in adults. Usual manifestations are headache and blurred vision. Sensitivity reactionsBecause sensitivity reactions are more likely to occur in persons with a history of allergy, hay fever, or urticaria, the preparation should be used with caution in such individuals. Cross-sensitization among the various tetracyclines is extremely common. OverdosageSymptomsNausea, vomiting, headache, increased intracranial pressure, skin pigmentation. Patient Information
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