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|Inamrinone Inamrinone |
Drugs search, click the first letter of a drug name: | A | B | C | D | E | F | G | H | I | J | K | L | M | N | O | P | Q | R | S | T | U | V | W | X | Y | Z | 1 | 2 | 3 | 4 | 5 | 6 | 8 | 9 Home InamrinonePronouncation: (in-AM-rih-nohn)Class: Inotropic agent Trade Names: Mechanism of ActionPharmacologyPositive inotropic agent with vasodilator activity. PharmacokineticsDistributionVd is 1.2 L/kg. 10 to 49% is protein bound. The t 1/2 is 4.6 min. MetabolismSeveral metabolites: N-glycolyl, N-acetate, O-glucaronide. EliminationThe t 1/2 is 3.6 hr. The primary route is via the urine. Peak10 minutes. Duration30 min to 2 hr (dose-dependent) Special PopulationsChildrenThere is increased Vd and decreased elimination t 1/2 . CHFIn CHF patients the mean elimination is t 1/2 of 5.8 hr. Monitor hemodynamic response or drug level. Indications and UsageShort-term management of CHF in patients whose condition can be closely monitored and who have not responded adequately to digitalis, diuretics, or vasodilators. ContraindicationsHypersensitivity to bisulfites. Dosage and AdministrationAdultsIV Initial dose: 0.75 mg/kg bolus slowly over 2 to 3 min. Maintenance: 5 to 10 mcg/kg/min; additional 0.75 mg/kg bolus may be given 30 min after initiating therapy, not to exceed total daily dose of 10 mg/kg. General Advice
Storage/StabilityProtect ampules from light. Store at room temperature. Drug InteractionsNone well documented. IncompatibilityChemical interaction occurs slowly over 24 hr when mixed directly with dextrose-containing solutions. Do not inject furosemide into IV line containing inamrinone; immediate precipitate forms. Laboratory Test InteractionsNone well documented. Adverse ReactionsCardiovascularArrhythmia; hypotension. GINausea; vomiting. HematologicThrombocytopenia. PrecautionsPregnancyCategory C . LactationUndetermined. ChildrenSafety and efficacy not established. Sulfite SensitivityMay cause allergic-type reaction in susceptible patients. ArrhythmiasSupraventricular and ventricular arrhythmias have occurred. Fluid balanceVigorous diuretic therapy may cause inadequate response to inamrinone therapy; liberalization of fluids may be needed. CVP monitoring has been advocated. HepatotoxicityDose may be reduced or drug may be discontinued if there are alterations in liver enzymes; if alterations occur with clinical symptoms, drug is discontinued. Post MINot recommended during acute phase. Severe aortic or pulmonic valvular diseaseNot recommended. ThrombocytopeniaMore common in patients on prolonged therapy. OverdosageSymptomsArrhythmias, excessive hypotension. Patient Information
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