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|Diazoxide, Oral |
Drugs search, click the first letter of a drug name: | A | B | C | D | E | F | G | H | I | J | K | L | M | N | O | P | Q | R | S | T | U | V | W | X | Y | Z | 1 | 2 | 3 | 4 | 5 | 6 | 8 | 9 Home Diazoxide, OralPronouncation: (DIE-aze-OX-ide)Class: Glucose-elevating agent Trade Names: Mechanism of ActionPharmacologyProduces prompt dose-related increase in blood glucose by inhibiting pancreatic insulin release. PharmacokineticsDistribution90% protein bound. Crosses the placenta. Eliminationt ½ is 24 to 36 hr. Excreted by kidneys. OnsetWithin 1 hr. DurationLess than 8 hr. Special PopulationsRenal Function Impairmentt ½ is prolonged. Indications and UsageManagement of hypoglycemia caused by hyperinsulinism in adults with inoperable islet cell adenoma or carcinoma or extrapancreatic malignancy, in infants and children with leucine sensitivity, islet cell hyperplasia, nesidioblastosis, extrapancreatic malignancy, islet cell adenoma or adenomatosis. ContraindicationsHypersensitivity to thiazides; functional hypoglycemia. Dosage and AdministrationAdults and ChildrenPO 3 to 8 mg/kg/day in 2 to 3 equal doses q 8 to 12 hr. Infants and NewbornsPO 8 to 15 mg/kg/day in 2 to 3 equal doses q 8 to 12 hr. Storage/StabilityStore at room temperature. Protect from light. Drug InteractionsAntihypertensive agentsEnhanced antihypertensive effect. HydantoinsPossible loss of seizure control. SulfonylureasDecreased pharmacologic effects of both drugs. Thiazide diureticsIncreased hyperglycemic and hyperuricemic effects of diazoxide; hypotension. Laboratory Test InteractionsHypoglycemia and hyperuricemia produced by diazoxide may affect assessment of these metabolic states. Increased renin secretion and IgG concentrations and decreased cortisol secretion may occur. False-negative insulin response to glucagon may occur. Adverse ReactionsCardiovascularTachycardia; palpitations; hypotension; transient hypertension; chest pain. CNSHeadache; weakness; malaise; anxiety; dizziness; insomnia; polyneuritis; paresthesia; extrapyramidal signs; fever. DermatologicHirsutism of lanugo type on forehead, back and limbs; skin rash; pruritus; monilial dermatitis; herpes; loss of scalp hair. EENTTransient cataracts; subconjunctival hemorrhage; ring scotoma; blurred vision; diplopia; lacrimation. GIAnorexia; nausea; vomiting; abdominal pain; ileus; diarrhea; transient loss of taste; acute pancreatitis; pancreatic necrosis. GenitourinaryAzotemia; decreased Ccr; reversible nephrotic syndrome; decreased urinary output; hematuria; albuminuria; glycosuria. HematologicThrombocytopenia with or without purpura; transient neutropenia; eosinophilia; decreased hemoglobin or hematocrit; excessive bleeding; decreased IgG. MetabolicHyperglycemia; increased serum uric acid; gout; galactorrhea; breast lump enlargement; increased AST and alkaline phosphatase. MiscellaneousSodium and fluid retention; advance in bone age. Precautions
PregnancyCategory C . LactationUndetermined. Labor and DeliveryMay cause cessation of uterine contractions. Renal FunctionMay have decreased protein binding of diazoxide resulting in increased hypotensive effect. Blood levelsMay be higher with liquid than with capsule formulation; use caution when changing dosage forms. Fluid retentionMay precipitate CHF in patients with compromised cardiac reserve. Ketoacidosis and nonketotic hyperosmolar comaMay occur with recommended doses. OverdosageSymptomsHypotension, hyperglycemia. Patient Information
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