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|Amobarbital Sodium |
Drugs search, click the first letter of a drug name: | A | B | C | D | E | F | G | H | I | J | K | L | M | N | O | P | Q | R | S | T | U | V | W | X | Y | Z | 1 | 2 | 3 | 4 | 5 | 6 | 8 | 9 Home Amobarbital SodiumPronouncation: (am-oh-BAR-bih-tahl SO-dee-uhm)Class: Sedative, Hypnotic, Barbiturate Trade Names: Mechanism of ActionPharmacologyDepresses sensory cortex; decreases motor activity; alters cerebellar function and produces drowsiness, sedation and hypnosis. PharmacokineticsDistributionRapidly distributed to all tissues and fluids, with high concentrations in brain, liver, and kidneys. Bound to plasma and tissue proteins. MetabolismMetabolized by hepatic microsomal enzyme system. EliminationPlasma t ½ is about 25 h. Metabolites excreted in urine and to a lesser extent in the feces. Negligible amount eliminated unchanged in urine. Onset0.75 to 1 h. Duration6 to 8 h. Indications and UsageRelief of anxiety; short-term therapy for insomnia; induction of preanesthetic sedation. ContraindicationsHypersensitivity to barbiturates; history of addiction to sedative-hypnotic drugs; history of porphyria; severe liver impairment; respiratory disease with dyspnea; patients with nephritis. Dosage and AdministrationInsomniaAdults PO/IM/IV 65 to 200 mg at bedtime. SedationAdults PO/IM/IV 30 to 50 mg twice daily or 3 times daily. ChildrenPO/IM 2 to 6 mg/kg/dose. General Advice
Storage/StabilityStore at room temperature. Do not freeze. Drug InteractionsAlcohol, CNS depressantsDepressant effects of these drugs may be enhanced. Anticoagulants, beta-blockers, calcium-channel blockers (eg, verapamil), theophyllinesActivity of these drugs may be reduced. AnticonvulsantsSerum concentrations of carbamazepine, valproic acid and succinimides may be reduced. Valproic acid may increase barbiturate serum levels. CorticosteroidsEffectiveness may be reduced. Estrogens, estrogen-containing oral contraceptivesEffectiveness may be reduced. Laboratory Test InteractionsDecreased serum bilirubin; false-positive phentolamine test results. Adverse ReactionsCardiovascularBradycardia; hypotension; syncope. CNSDrowsiness; agitation; confusion; headache; hyperkinesia; ataxia; CNS depression; paradoxical excitement; nightmares; psychiatric disturbances; hallucinations; insomnia; dizziness. GINausea; vomiting; constipation. HematologicBlood dyscrasias (agranulocytosis, thrombocytopenia). HepaticLiver damage. RespiratoryHypoventilation; apnea; laryngospasm; bronchospasm. MiscellaneousHypersensitivity reactions (eg, angioedema, rashes, exfoliative dermatitis); fever; injection site reactions (eg, local pain, thrombophlebitis). Precautions
PregnancyCategory D . LactationExcreted in breast milk. ChildrenSafety and efficacy not established in children younger than 6 yr of age. ElderlyReduce dosage. Renal FunctionUse with caution; reduce dosage. Hepatic FunctionUse with caution; reduce dosage. Drug dependenceTolerance or psychologic and physical dependence may occur with continued use. OverdosageSymptomsRespiratory depression, CNS depression progressing to Cheyne-Stokes respiration, oliguria, tachycardia, hypotension, hypothermia, coma, shock, cessation of electrical activity in brain (extreme overdose). Patient Information
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